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配伍选择题 分子内有氨基甲酸酯结构,可以选择性地抑制MAO-A活性,阻断5-HT和NA的代谢的抗抑郁药是
A A B B C C D D E E F F G H
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配伍选择题 分子中的三氟甲基对选择性5-HT再摄取的亲和力和选择性起关键作用;分子中含C=N双键,只有E-异构体有活性的非三环类的抗抑郁药是
A A B B C C D D E E F F G H
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配伍选择题 结构中含有吗啉结构和酰胺结构,对MAO-A有可逆性抑制作用,从而提高脑内去甲肾上腺素、多巴胺和5-羟色胺的水平,产生抗抑郁作用的药物是
A A B B C C D D E E F F G H
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配伍选择题 本身无活性,必需先在肝内转化后才有效的药物是
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248933_0.png"> B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248933_0_1.png"> C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248933_0_2.png"> D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248933_0_3.png"> E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248933_0_4.png">
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配伍选择题 系21位酯化衍生物,由于全身性吸收作用,可造成可逆性下丘脑-垂体-肾上腺轴的抑制,部分患者可出现库欣综合征、高血糖等,所以只能外用的药物是
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248934_0.png"> B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248934_0_1.png"> C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248934_0_2.png"> D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248934_0_3.png"> E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248934_0_4.png">
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配伍选择题 可看成依那普利结构中的脯氨酸被八氢-1H-吲哚羧酸所替代的药物
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248938_0.png">图1 B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248938_0_1.png">图2 C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248938_0_2.png">图3 D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248938_0_3.png">图4 E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248938_0_4.png">图5
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配伍选择题 结构中有戊酸取代、脯氨酸被八氢-1H-吲哚羧酸替代的药物
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248939_0.png">图1 B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248939_0_1.png">图2 C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248939_0_2.png">图3 D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248939_0_3.png">图4 E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248939_0_4.png">图5
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配伍选择题 含有二羟基四氢萘的苯丙醇胺结构的非选择性β受体阻断药是
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248940_0.png">图1 B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248940_0_1.png">图2 C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248940_0_2.png">图3 D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248940_0_3.png">图4 E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248940_0_4.png">图5
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配伍选择题 含有吗啉取代噻二唑基的芳氧丙醇胺类非选择性β受体阻断药是
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248941_0.png">图1 B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248941_0_1.png">图2 C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248941_0_2.png">图3 D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248941_0_3.png">图4 E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248941_0_4.png">图5
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配伍选择题 具有苯丙醇胺结构和烯丙基结构的非选择性β受体阻断药是
A <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248942_0.png">图1 B <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248942_0_1.png">图2 C <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248942_0_2.png">图3 D <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248942_0_3.png">图4 E <img border="0" alt="" src="https://tuku.weimei168.com/uploads/upimg/20260227/24248942_0_4.png">图5
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